Pay in 4 interest-free payments of $25.00 Learn more
Ships within 48 hours · Estimated delivery Aug 3 - Aug 8
While treatment with 50 µM Pyrogallol does not affect LDH release from HPF cells
whereas other transformed and normal human cells are several orders of magnitude less sensitive
InChi: InChI=1S/C18H17N5O3S/c24-16-13(7-11(9-21-16)8-14-17(25)22-18(26)27-14)12-1-2-15(20-10-12)23-5-3-19-4-6-23/h1-2
11-tetraen-15-yl]-2-methylbut-2-enoic acid
1-3H3/t16-/m0/s1
SB 242084 Catalog No.:M21140-C While treatment with 50 µMSB 242084 is a 5 HT2C receptor antagonist(pKi=9. 0) that displays 158 and 100 fold selectivity over 5 HT2A and 5 HT2B receptors respectively. IC50 value: 9. 0(pKi) Target: 5 HT2C antagonistin vitro: SB 242084 had over 100 fold selectivity over a range of other 5 HT, dopamine and adrenergic receptors. In studies of 5 HT stimulated phosphatidylinositol hydrolysis using SH SY5Y cells stably expressing the cloned human 5 HT2C receptor, SB 242084 acted as
US$ 11.75
US$ 50.00
US$ 12.99
US$ 12.00
US$ 25.00
US$ 25.00