Dynorphin A (1-8) 8021 Smiles: CC1=C(C=C2SC(=O)N(C3C=CC=CC=3)C2=O)C=C(C)N1C1=CN=CC=C1

Smiles: CC1=C(C=C2SC(=O)N(C3C=CC=CC=3)C2=O)C=C(C)N1C1=CN=CC=C1

100 and 150 mg/kg

TBPB displays unprecedented functional selectivity at the M₁ mAChR

Smiles: COC1C=C2O[C@H]3[C@H](COC4=CC(O)=CC=C43)C2=CC=1

Smiles: CC1=CC(O)=C2C(=C1)C(=O)C1=CC=CC(O[C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)=C1C2=O

Dynorphin A (1-8) 8021 Smiles: CC1=C(C=C2SC(=O)N(C3C=CC=CC=3)C2=O)C=C(C)N1C1=CN=CC=C1Dynorphin A (1 8) is the predominant opioid peptide identified in placental tissue extracts. Dynorphin A (1 8) is the most likely natural ligand of the kappa receptor. The binding of 3H Bremazocine to the purified kappa receptor is inhibited by Dynorphin A (1 8) (IC50=303 nM). Product information CAS Number: 75790 53 3 Molecular Weight: 981. 15 Formula: C46H72N14O10 Chemical Name: (2S,3S) 2 [(2S) 2 [(2S) 2 [(2S) 2 [(2S) 2 (2 {2 [(2S) 2 amino 3 (4