Nalfurafine 061PEG17-Hydrazide 18-13)19-20-15/h8-13

18-13)19-20-15/h8-13

with IC50 of 5 nM (HTRF binding assays) and 20 nM (MTT proliferation assays)

Formula: C19H22Cl2N4

highly potent and selective histamine H1-receptor antagonist with anti-allergic activity

Chemical Name: ethyl N-[(2S)-5-amino-2-methyl-3-phenyl-1H

Nalfurafine 061PEG17-Hydrazide 18-13)19-20-15/h8-13Nalfurafine (TRK 820) is a potent selective and orally active G protein biased kappa opioid receptor (KOR) agonist with high translational potential. Nalfurafine (TRK 820) enhances the therapeutic potential of MOR targeting analgesics, has the potential for uremic pruritis treatment. Product information CAS Number: 152657 84 6 Molecular Weight: 476. 56 Formula: C28H32N2O5 Chemical Name: (2E) N [(1S,5R,13R,14R,17S) 4 (cyclopropylmethyl) 10,17 dihydroxy