TG4-155 62175 also known as Branaplam and

also known as Branaplam and LMI-070

Chemical Name: (4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluoromethyl)-2

23)24/h9-12

Chen (Leguminosae)

Solubility: DMSO : 2 mg/mL (9

TG4-155 62175 also known as Branaplam andTG4 155 is a potent, brain permeant and selective EP2 receptor antagonist with a Ki of 9. 9 nM. TG4 155 shows low nanomolar antagonist activity against only EP2 and DP1. TG4 155 has an EP2 Schild KB of 2. 4 nM and displays 550 4750 fold selectivity for EP2 over EP1, EP3, EP4 and IP, but only 14 fold selectivity against the DP1 receptor. Product information CAS Number: 1164462 05 8 Molecular Weight: 394. 46 Formula: C23H26N2O4 Chemical Name: (2E) N [2